- 中間體
- 酒石酸伐尼克蘭 230615-70-0
- 阿瑞匹坦 287930-73-8
- 阿瑞匹坦 127852-28-2
- 阿瑞匹坦 287930-75-0
- 阿瑞匹坦 200000-59-5
- 阿瑞匹坦 155742-64-6
- 阿瑞匹坦 252742-72-6
- 福沙匹坦雙葡甲胺 990-91-0
- 福沙匹坦雙葡甲胺 265121-01-5
- 維格列汀 207557-35-5
- 維格列汀 702-82-9
- 艾氟康唑 144230-50-2
- 艾氟康唑 133775-25-4
- 艾氟康唑 127000-90-2
- 釓特酸葡胺
- 米拉貝隆
- 盧立康唑 98873-55-3
- 盧立康唑 126534-31-4
- 硫酸阿扎那韋
- 硼替佐米 179324-87-9
- 硼替佐米 114457-94-2
- 硼替佐米 205393-22-2
- 布林佐胺
- 利伐沙 446292-08-6
- 利伐沙 446292-07-5
- 西那卡塞 1005450-55-4
- 西那卡塞 585-50-2
- 依來曲普坦 585-50-2
- 茚達特羅 312753-53-0
- 茚達特羅 173140-90-4
- 西他列汀
- 福沙那韋鈣
熱門資訊
中間體
中间体
- 分類:中間體
- 發佈時間:2020-03-11 00:00:00
- 訪問量:0
概要:
詳情
對應API | CAS | Structure | KSM/Interm. | Chemical Name | US DMF | |
1 | 酒石酸伐尼克蘭 Varenicline Tartrate |
230615-70-0 | Interm | 2,2,2 - trifluoro - 1 - (6,7,9,10-tetrahydro- 8H - 6,10 -methanoazepino [4,5-g]quinoxaline- 8 - yl) ethan - 1 - one | Tech Pack | |
2 | 阿瑞匹坦 Aprepitant |
287930-73-8 | KSM | 4-Benzyl-2-hydroxy-morpholin-3-one | Tech Pack | |
127852-28-2 | KSM | (1R)-1-[3,5-Bis(trifluoromethyl) phenyl]ethanol | Tech Pack | |||
287930-75-0 | Interm | (R)-2-((R)-1-(3,5-bis (trifluoromethyl)phenyl) ethoxy)-4-benzylmorpholin-3-one |
Tech Pack | |||
200000-59-5 | Interm | (2R, 3S)-2-[(1R)-l-[3, 5-Bis (trifluoromethyl)phenyl] ethoxy]-3-(4-fluorophenyl) morpholine, 4- methylbenzenesulfonate | √ | |||
155742-64-6 | Interm | N-Methylcarbonyl-2-chloroacetamidrazone | Tech Pack | |||
252742-72-6 | Interm | 5-Chloromethyl-2,4-Dithydro-[1,2,4]Triazol-3-One | Tech Pack | |||
3 | 福沙匹坦雙葡甲胺 Fosaprepitant Dimeglumine |
990-91-0 | Interm | Tetrabenzyl pyrophosphate | Tech Pack | |
265121-01-5 | Interm | Dibenzyl (3-(((2R,3S)-2-((R)-1-(3,5-bis(trifluoromethyl)phenyl)ethoxy)-3-(4-fluorophenyl)morpholino)methyl)-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)phosphonate | Tech Pack | |||
4 | 維格列汀 Vildagliptin |
207557-35-5 | Interm | (S)-1-(2-chloroacetyl)pyrrolidine-2- carbonitrile |
Tech Pack | |
702-82-9 | Interm | 3-Amino-1-hydroxyadamantane | Tech Pack | |||
5 | 艾氟康唑 Efinaconazole |
144230-50-2 | Interm | 4-Methylidenepiperidine, hydrochloride | Tech Pack | |
133775-25-4 | Interm | (2R,3R)-2-(2,4-difluorophenyl)-1-(1H-1,2,4-triazol-1-yl)butane-2,3-diol | √ | |||
127000-90-2 | Interm | 1-(((2R,3S)-2-(2,4-difluorophenyl)-3-methyloxiran-2-yl)methyl)-1H-1,2,4-triazole | √ | |||
6 | 釓特酸葡胺 Gadoterate Meglumine |
60239-18-1 | Interm | 1,4,7,10-tetraazacyclododecane-1,4,7,10-tetraacetic acid | Tech Pack | |
7 | 米拉貝隆 Mirabegron |
20780-53-4 | Interm | (R)-Styrene oxide | Tech Pack | |
8 | 盧立康唑 Luliconazole |
98873-55-3 | Interm | Imidazole-1-yl-acetonitrile | Tech Pack | |
126534-31-4 | Interm | (S)-2-chloro-1-(2,4-dich lorophenyl) ethanol |
Tech Pack | |||
9 | 硫酸阿扎那韋 Atazanavir sulfate |
198904-86-8 | Interm | 2-[(2S,3S)-3-[[(1,1-Dimethylethoxy) carbonyl]amino]-2-hydroxy-4-phenyl-butyl]-2-[[4-(2-pyridinyl)phenyl] methyl] hydrazinecarboxylic acid, 1,1-dimethylethyl ester | Tech Pack | |
10 |
硼替佐米 Bortezomib |
179324-87-9 | Interm | (aR,3aS,4S,6S,7aR)-Hexahydro-3a,8,8-trimethyl-alpha-(2-methylpropyl)-4,6-methano-1,3,2-benzodioxaborole-2-methanamine 2,2,2-trifluoroacetate | Tech Pack | |
114457-94-2 | Interm | N-(2-Pyrazinylcarbonyl)-L-phenylalanine | Tech Pack | |||
205393-22-2 | Interm | Bortezomib pinanediol ester | Tech Pack | |||
11 |
布林佐胺 Brinzolamide |
160982-16-1 | Interm | (S)-3,4-Dihydro-6-chloro-4-hydroxy-4H-thieno[3,2-e]-1,2-thiazine-1,1-dioxide | Tech Pack | |
12 |
利伐沙 Rivaroxaban |
446292-08-6 | Interm | 2-[[(5S)-2-Oxo-3-[4-(3-oxo-4-morpholinyl)phenyl]-5-oxazolidinyl] methyl]-1H-isoindole-1,3(2H)-dione | Tech Pack | |
446292-07-5 | Interm | 2-[(2R)-2-Hydroxy-3-[[4-(3-oxo-4-morpholinyl)-phenyl]amino]propyl]-1H-isoindole-1,3(2H)-dione | Tech Pack | |||
13 |
西那卡塞 Cinacalcet |
1005450-55-4 | Interm | N-((R)-1-(naphthalen-1-yl)ethyl)-3-(3-(trifluoromethyl)phenyl)-propanamide | Tech Pack | |
585-50-2 | Interm | 3-(3-Trifluoromethylphenyl)propionic acid | Tech Pack | |||
14 |
依來曲普坦 Eletriptan |
143322-57-0 | Interm | (R)-5-Bromo-3-((1-methylpyrrolidin-2-yl)methyl)-1H-indole | Tech Pack | |
15 |
茚達特羅 Indacaterol |
312753-53-0 | Interm | 5,6-Diethyl-2,3-dihydro-1H-inden-2-amine hydrochloride | Tech Pack | |
173140-90-4 | Interm | 5-(2R)-2-Oxiranyl-8-benzyloxy-2(1H)-quinolinone | Tech Pack | |||
16 |
西他列汀 Sitagliptin |
764667-65-4 | Interm | (2Z)-4-Oxo-4-[3-(trifluoromethyl)-5,6-dihydro-[1,2,4]triazolo[4,3-a]-pyrazine-7(8H)-yl]-1-(2,4,5-trifluorophenyl)butan-2-one | Tech Pack | |
17 | 福沙那韋鈣Fosamprenavir calcium | 160232-08-6 | Interm | ([1S,2R]-(1-Benzyl-2-hydroxy-3-(isobutyl-amino)-propyl)carbamic acid tert-butylester | Tech Pack | |
18 | 878376-35-3 | KSM | Pyridine-2-sulfonyl fluoride | Tech Pack | ||
19 | 473923-95-4 | KSM | 3-Fluoro-5-hydroxybenzonitrile | Tech Pack |
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